SCHEMBL11679062

SCHEMBL11679062

O=C(O)CNC(=O)Nc1ncnc2nc[nH]c12

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 8/20 0.58
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
NT5C2 P49902 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.52
TSHR P16473 2/20 0.51
TP53 P04637 1/20 0.51
HSD17B10 Q99714 1/20 0.51
NT5E P21589 1/20 0.51
BRAF P15056 2/20 0.50
CYP3A4 P08684 1/20 0.50
TOP2A P11388 1/20 0.50
CYP1A2 P05177 2/20 0.49
HIF1A Q16665 1/20 0.49
LMNA P02545 1/20 0.47
CYP2D6 P10635 1/20 0.47
CDK2 P24941 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15709153 0.82 TSHR (0.67) BRD4SMN1; SMN2TSHRTP53HSD17B10
SCHEMBL30919395 0.82 TSHR (0.67) BRD4SMN1; SMN2TSHRTP53HSD17B10
SCHEMBL22118772 0.81 BRD4 (0.68) BRD4NPC1RAB9ANT5C2SMN1; SMN2
SCHEMBL19466078 0.80 NPC1 (0.54) BRD4NPC1RAB9ANT5C2SMN1; SMN2
SCHEMBL28669706 0.80 NPC1 (0.63) BRD4NPC1RAB9ANT5C2SMN1; SMN2
SCHEMBL3038563 0.78 NPC1 (0.76) BRD4NPC1RAB9ANT5C2SMN1; SMN2
SCHEMBL29638098 0.77 NPC1 (0.56) BRD4NPC1RAB9ANT5C2SMN1; SMN2
SCHEMBL17372610 0.77 NPC1 (0.56) BRD4NPC1RAB9ANT5C2SMN1; SMN2
SCHEMBL28828155 0.77 BRD4 (0.59) BRD4NPC1RAB9ANT5C2SMN1; SMN2
SCHEMBL9853721 0.76 SMN1; SMN2 (0.60) BRD4NT5C2SMN1; SMN2TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4038480-A HYPOTENSIVE AGENTS;INCREASE CARDIAC OUTPUT;ENZYME ACTIVATORS ICN PHARMACEUTICALS, INC. (US) 1977-07-26 US disclosed