SCHEMBL9853810

SCHEMBL9853810

COc1ccc(Oc2cnccc2N)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.54
PTGS2 P35354 4/20 0.54
CYP3A4 P08684 4/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
RAB9A P51151 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
IKBKB O14920 1/20 0.43
ALDH1A1 P00352 4/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
MAPK1 P28482 1/20 0.42
ICAM1 P05362 1/20 0.42
SELE P16581 1/20 0.42
CCNC P24863 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7054411 0.86 TEAD4 (0.47) PTGS1PTGS2CYP3A4CYP1A2CYP2D6
SCHEMBL4370948 0.82 PTGS1 (0.52) PTGS1PTGS2CYP3A4CYP1A2CYP2D6
SCHEMBL4370679 0.82 PTGS1 (0.52) PTGS1PTGS2CYP3A4CYP1A2CYP2D6
SCHEMBL4374807 0.81 PTGS1 (0.50) PTGS1PTGS2CYP3A4CYP1A2CYP2C9
SCHEMBL9853800 0.81 MAPT (0.50) PTGS1PTGS2CYP3A4CYP1A2CYP2D6
SCHEMBL222945 0.81
SCHEMBL31576017 0.81
Hydrochloric Acid SCHEMBL9853816 0.80 PTGS1 (0.49) PTGS1PTGS2CYP3A4CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL29374919 0.79 CA12 (0.47) PTGS1CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL1282569 0.79 GAA (0.38) PTGS1PTGS2CYP3A4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4959377-A Phenoxypyridinamine compounds which are use as a dermatological composition HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-09-25 US claimed
EP-0405487-A1 Phenoxypyridinamines and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-02 EP disclosed
US-4959377-A Phenoxypyridinamine compounds which are use as a dermatological composition HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-09-25 US disclosed