SCHEMBL9853906

SCHEMBL9853906

N#Cc1cc(C(=O)CO)ccc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39
GSK3B P49841 2/20 0.36
ALDH1A1 P00352 3/20 0.35
HPGD P15428 1/20 0.35
MAPT P10636 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
XDH P47989 1/20 0.34
HSP90AA1 P07900 1/20 0.33
NTSR1 P30989 1/20 0.33
USP2 O75604 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29896948 0.85 GSK3B (0.54) MAPK1CYP1A2CYP3A4TSHRADRB2
SCHEMBL10493941 0.85 GSK3B (0.43) MAPK1CYP1A2CYP3A4TSHRADRB2
SCHEMBL5165644 0.85 GSK3B (0.54) MAPK1CYP1A2CYP3A4TSHRADRB2
SCHEMBL13974083 0.85 PGR (0.42) MAPK1CYP1A2CYP3A4TSHRADRB2
SCHEMBL9821246 0.85 MAPK1 (0.38) MAPK1CYP1A2CYP3A4TSHRADRB2
SCHEMBL5070972 0.82 MAPK1 (0.43) MAPK1CYP1A2CYP3A4TSHRADRB2
SCHEMBL4026182 0.80 CDC25B (0.50) TSHRALDH1A1HPGDMAPTTDP1
SCHEMBL6816025 0.80 PARP15 (0.43) MAPK1CYP1A2CYP3A4TSHRADRB2
SCHEMBL8060674 0.79 VNN1 (0.45) TSHRGSK3BALDH1A1NPC1
SCHEMBL23302174 0.79 TSHR (0.38) MAPK1CYP1A2CYP3A4TSHRADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5071871-A Pharmaceutically useful benzo(β)pyranes and pyranopyridines SANDOZ LTD. (CH) 1991-12-10 US disclosed
EP-0439054-A1 Monoazo dyes, their preparation and use CASSELLA Aktiengesellschaft (DE) 1991-07-31 EP disclosed
US-RE32196-E PROPHYLACTIC CHEMOTHERAPY OF ALLERGIC CONDITIONS LILLY INDUSTRIES LIMITED (GB) 1986-07-01 US disclosed
EP-0038615-A2 Disperse monoazo dyes IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1981-10-28 EP disclosed