SCHEMBL9854835

SCHEMBL9854835

CCCC1CC=C(C#Cc2ccc(-c3ccc(C#N)cc3F)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 13/20 0.41
DRD3 P35462 2/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
MAOB P27338 1/20 0.32
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9856043 0.94 KDM1A (0.40) KDM1ADRD3DRD2DRD4CYP11B1
SCHEMBL9854880 0.93 KDM1A (0.39) KDM1ADRD3DRD2DRD4CYP11B1
SCHEMBL9855144 0.92 KDM1A (0.39) KDM1ADRD3DRD2DRD4CYP11B1
SCHEMBL9855680 0.91 KDM1A (0.40) KDM1ADRD3DRD2DRD4CYP11B1
SCHEMBL9855095 0.87 DRD2 (0.38) KDM1ADRD3DRD2DRD4
SCHEMBL9855747 0.86 DRD3 (0.43) KDM1ADRD3DRD2DRD4MAOB
SCHEMBL9854848 0.86 DRD2 (0.37) KDM1ADRD3DRD2DRD4
SCHEMBL9855303 0.85 RARB (0.38) KDM1ADRD3DRD2DRD4
SCHEMBL9855498 0.84 RARB (0.41) KDM1ADRD3DRD2DRD4
SCHEMBL10509821 0.82 DRD3 (0.40) KDM1ADRD3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed
EP-0306505-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES. MERCK PATENT GMBH (DE) 1989-03-15 EP disclosed
WO-1988007523-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-06 WO disclosed