SCHEMBL9854974

SCHEMBL9854974

Cc1ccc(S(=O)(=O)OC2CCN(C(=O)OCc3ccc([N+](=O)[O-])cc3)C2)cc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
MAPT P10636 3/20 0.47
HPGD P15428 1/20 0.47
KDM4E B2RXH2 1/20 0.46
CYP2D6 P10635 1/20 0.45
GRIN2B Q13224 3/20 0.43
F2 P00734 1/20 0.43
NPC1 O15118 1/20 0.42
KMT2A Q03164 1/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10639380 0.94 KDM4E (0.49) ALDH1A1MAPTHPGDKDM4ECYP2D6
SCHEMBL24064971 0.90 SMN1; SMN2 (0.48) ALDH1A1MAPTKDM4ENPC1KMT2A
SCHEMBL5723831 0.87 ALDH1A1 (0.45) ALDH1A1MAPTHPGDKDM4ENPC1
SCHEMBL5723815 0.87 ALDH1A1 (0.45) ALDH1A1MAPTHPGDKDM4ENPC1
SCHEMBL3789109 0.87 SMN1; SMN2 (0.51) MAPTCYP2D6GRIN2BNPC1LMNA
SCHEMBL3615713 0.87 SMN1; SMN2 (0.51) MAPTCYP2D6GRIN2BNPC1LMNA
SCHEMBL8788495 0.87 SMN1; SMN2 (0.51) MAPTCYP2D6GRIN2BNPC1LMNA
SCHEMBL10639596 0.83 GRIN2B (0.56) ALDH1A1MAPTHPGDKDM4EGRIN2B
SCHEMBL6767786 0.82 KDM4E (0.43) ALDH1A1MAPTKDM4ENPC1LMNA
SCHEMBL5724304 0.81 ALDH1A1 (0.47) ALDH1A1MAPTHPGDKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5071843-A Thienamycin antibiotics with delayed metabolism MERCK & CO., INC. (US) 1991-12-10 US disclosed
EP-0161541-B1 6-[1-Hydroxyethyl]-2-SR8-1-methyl-1-carba-dethiapen-2-em-3-carboxylic acids MERCK & CO. INC. (US) 1990-12-12 EP disclosed
EP-0161546-B1 COMBINATION OF 2-SUBSTITUTED CARBAPENEMS WITH DIPEPTIDASE INHIBITORS MERCK & CO. INC. (US) 1989-12-13 EP disclosed
US-4696923-A THIENAMYCIN ANTIBIOTICS, BACTERICIDES MERCK & CO., INC. (US) 1987-09-29 US disclosed
EP-0161546-A1 Combination of 2-substituted carbapenems with dipeptidase inhibitors MERCK & CO. INC. (US) 1985-11-21 EP disclosed
EP-0161541-A1 6-[1-Hydroxyethyl]-2-SR8-1-methyl-1-carba-dethiapen-2-em-3-carboxylic acids MERCK & CO. INC. (US) 1985-11-21 EP disclosed