SCHEMBL985675

SCHEMBL985675

Nc1ncc(C2=CCN(C(=O)O)CC2)cc1-c1nnnn1-c1cccc(F)c1F

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 5/20 0.37
CDK9 P50750 5/20 0.37
KCNN4 O15554 5/20 0.37
GRM1 Q13255 7/20 0.36
GRM5 P41594 5/20 0.36
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
HRH1 P35367 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL987228 0.96 KCNN4 (0.35) CCNT1CDK9KCNN4GRM1GRM5
SCHEMBL988378 0.92 ERN1 (0.40) CCNT1CDK9KCNN4GRM1GRM5
SCHEMBL987001 0.91 ALDH1A1 (0.38) CCNT1CDK9KCNN4GRM1GRM5
SCHEMBL986695 0.90 NAMPT (0.41) CCNT1CDK9KCNN4GRM1GRM5
SCHEMBL982752 0.90 GRM1 (0.39) CCNT1CDK9KCNN4GRM1GRM5
SCHEMBL985805 0.90 NAMPT (0.39) CCNT1CDK9KCNN4GRM1GRM5
SCHEMBL984594 0.89 ERN1 (0.37) CCNT1CDK9KCNN4GRM1GRM5
SCHEMBL987033 0.88 CDK9 (0.39) CCNT1CDK9KCNN4GRM1GRM5
SCHEMBL2076538 0.88 GRM5 (0.51) CCNT1CDK9GRM1GRM5
SCHEMBL984990 0.88 NAMPT (0.38) CCNT1CDK9KCNN4GRM1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7872031-B2 c-MET protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-01-18 US claimed