SCHEMBL9857433

SCHEMBL9857433

CCCCCCCOc1cccc(C(=O)Nc2ccccc2OCc2nnn[nH]2)c1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 3/20 0.52
NR1H4 Q96RI1 3/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
TP53 P04637 1/20 0.49
POLB P06746 1/20 0.49
THRB P10828 1/20 0.48
CYSLTR2 Q9NS75 1/20 0.48
CYSLTR1 Q9Y271 1/20 0.48
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48
TSHR P16473 1/20 0.48
PLK1 P53350 1/20 0.47
PTPN1 P18031 2/20 0.46
KAT6A Q92794 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713817 0.90 PLK1 (0.59) CYSLTR2CYSLTR1PLK1
SCHEMBL9857033 0.88 NR1H4 (0.63) SMPD1NR1H4MEN1KMT2ATHRB
SCHEMBL9132501 0.87 PLK1 (0.52) NR1H4CYSLTR2CYSLTR1PLK1
SCHEMBL9132741 0.87 PLK1 (0.52) NR1H4CYSLTR2CYSLTR1PLK1
SCHEMBL10721101 0.82 NR1H4 (0.59) NR1H4MEN1KMT2ATP53THRB
SCHEMBL9713298 0.81 SMPD1 (0.60) SMPD1NR1H4MEN1KMT2ATP53
SCHEMBL9135604 0.80 CACNA1H (0.49) NR1H4CYSLTR2CYSLTR1PLK1
SCHEMBL9255356 0.79 PLK1 (0.44) MEN1KMT2ACYSLTR2CYSLTR1PLK1
SCHEMBL9254816 0.79 PLK1 (0.44) MEN1KMT2ACYSLTR2CYSLTR1PLK1
SCHEMBL9254823 0.78 CYSLTR2 (0.52) MEN1KMT2ACYSLTR2CYSLTR1PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994479-A Antagonists of SRS-A(slow reacting substance of anaphylaxis); antiallergens, antiischemic agents YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-02-19 US disclosed
EP-0218728-A1 PHENYLENE DERIVATIVES YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1987-04-22 EP disclosed
WO-1986005779-A1 PHENYLENE DERIVATIVES YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1986-10-09 WO disclosed