SCHEMBL9857528

SCHEMBL9857528

CC[S+]([O-])CCC(=O)NN

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.52
KDM4E B2RXH2 2/20 0.41
KDM5C P41229 1/20 0.41
PHF8 Q9UPP1 1/20 0.41
KDM2A Q9Y2K7 1/20 0.41
ALDH1A1 P00352 2/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
MAPT P10636 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
GAA P10253 2/20 0.32
CYP2D6 P10635 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19667831 0.87 KDM4E (0.48) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL7749331 0.78
SCHEMBL9325348 0.73
SCHEMBL17038880 0.73
SCHEMBL8257596 0.72 TSHR (0.50) KDM4EALDH1A1POLBHTTMAPT
SCHEMBL11249999 0.71
Dimethyl Sulfoxide SCHEMBL28118530 0.71 CTSD (0.52) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL9857497 0.71 CTSD (0.46) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL19682728 0.69 CTSD (0.41) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL924945 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0193822-B1 8-Chlorodibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid, 2-(thio-, sulfinyl- and sulfonyl-containing acyl)hydrazides G.D. Searle & Co. (US) 1991-03-20 EP claimed
EP-0193822-A2 8-Chlorodibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid, 2-(thio-, sulfinyl- and sulfonyl-containing acyl)hydrazides G.D. Searle & Co. (US) 1986-09-10 EP claimed
US-4559336-A 8-Chlorodibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid, 2-(sulfinyl- and sulfonyl-containing acyl)hydrazides G.D. SEARLE & CO. (US) 1985-12-17 US claimed
US-4614617-A Intermediates for 8-chlorodibenz[(b,f)][1,4]oxazepine-10(11H)-carboxylic acid, 2-(sulfinyl- and sulfonyl-containing acyl)hydrazides G. D. SEARLE & CO. (US) 1986-09-30 US disclosed
US-4559336-A 8-Chlorodibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid, 2-(sulfinyl- and sulfonyl-containing acyl)hydrazides G.D. SEARLE & CO. (US) 1985-12-17 US disclosed