SCHEMBL9857552

SCHEMBL9857552

O=C1C(O)=C(C2CCC(c3ccccc3)CC2)C(=O)c2ccccc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.62
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
USP2 O75604 1/20 0.62
LMNA P02545 1/20 0.62
TP53 P04637 1/20 0.62
CYP1A2 P05177 1/20 0.62
CYP2C9 P11712 1/20 0.62
HPGD P15428 1/20 0.62
TSHR P16473 1/20 0.62
HIF1A Q16665 1/20 0.62
APAF1 O14727 1/20 0.48
TDP2 O95551 1/20 0.48
ALDH1A1 P00352 4/20 0.42
MAPK10 P53779 1/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C1 Q04828 1/20 0.41
P2RX7 Q99572 3/20 0.41
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Atovaquone SCHEMBL20769805 0.88 MAPT (0.82) MAPTMEN1KMT2AUSP2LMNA
SCHEMBL15305631 0.88 MEN1 (0.60) MAPTMEN1KMT2AUSP2LMNA
Atovaquone SCHEMBL21694 0.88 MAPT (0.82) MAPTMEN1KMT2AUSP2LMNA
Atovaquone SCHEMBL637069 0.88 MAPT (0.82) MAPTMEN1KMT2AUSP2LMNA
Atovaquone SCHEMBL8848607 0.88 MAPT (0.82) MAPTMEN1KMT2AUSP2LMNA
Atovaquone SCHEMBL29559044 0.88 MAPT (0.82) MAPTMEN1KMT2AUSP2LMNA
Atovaquone SCHEMBL1542719 0.88 MAPT (0.82) MAPTMEN1KMT2AUSP2LMNA
Atovaquone SCHEMBL9975142 0.88 MAPT (0.82) MAPTMEN1KMT2AUSP2LMNA
SCHEMBL8610391 0.88 MAPT (0.50) MAPTMEN1KMT2AUSP2LMNA
SCHEMBL9857346 0.84 APAF1 (0.54) MAPTMEN1KMT2AUSP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5053418-A Synergistic mixture of 2-(4,-(4-chlorophenyl)cyclohexyl)3-hydr oxy-1,4 napthoquinone and 3,5-dichloro-2,6 dichloropyridinol BURROUGHS WELLCOME CO. (US) 1991-10-01 US disclosed
EP-0123239-B1 IMPROVEMENTS IN OR RELATING TO ANTIPROTOZOAL AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-11 EP disclosed
EP-0401875-A2 Improvements in or relating to antiprotozoal agents THE WELLCOME FOUNDATION LIMITED (GB) 1990-12-12 EP disclosed