SCHEMBL9858008

SCHEMBL9858008

O=C(O)c1cn(Cc2c(F)cccc2Cl)nn1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.65
CA5A P35218 1/20 0.64
LMNA P02545 3/20 0.63
ALDH1A1 P00352 3/20 0.63
KLKB1 P03952 1/20 0.45
EGFR P00533 1/20 0.44
KDM4E B2RXH2 2/20 0.44
DPP4 P27487 1/20 0.43
PRSS12 P56730 1/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 1/20 0.42
SLC22A12 Q96S37 1/20 0.42
ALKBH1 Q13686 1/20 0.42
RORC P51449 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL460913 0.90 CA5A (0.76) CYP2C19CA5ALMNAALDH1A1KLKB1
SCHEMBL9857399 0.88 CA5A (0.82) CYP2C19CA5ALMNAALDH1A1KLKB1
SCHEMBL9858012 0.81 CYP2C19 (0.56) CYP2C19CA5ALMNAALDH1A1EGFR
SCHEMBL460954 0.81 CA5A (0.74) CYP2C19CA5ALMNAALDH1A1KLKB1
SCHEMBL10664054 0.78 CA5A (0.70) CYP2C19CA5ALMNAALDH1A1KLKB1
SCHEMBL10662617 0.78 TYR (0.53) CYP2C19LMNAALDH1A1KMT2AMEN1
Rufinamide SCHEMBL230448 0.78 CA5A (1.00) CYP2C19CA5ALMNAALDH1A1KLKB1
SCHEMBL9858144 0.78 CA5A (0.55) CA5ALMNAALDH1A1DPP4KMT2A
Rufinamide SCHEMBL20769779 0.78 CA5A (1.00) CYP2C19CA5ALMNAALDH1A1KLKB1
SCHEMBL6738882 0.78 CA5A (0.74) CYP2C19CA5ALMNAALDH1A1KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP disclosed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US disclosed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP disclosed