SCHEMBL9858151

SCHEMBL9858151

COc1c(C(N)=O)sc2ccc(C(F)(F)F)cc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICAM1 P05362 5/20 0.54
SELE P16581 5/20 0.54
VCAM1 P19320 1/20 0.54
PRNP P04156 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
PPARG P37231 1/20 0.43
HTT P42858 1/20 0.43
MAPK10 P53779 1/20 0.43
NCOA2 Q15596 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
CSNK1D P48730 3/20 0.41
CFTR P13569 1/20 0.40
AGPAT2 O15120 1/20 0.39
CISD2 Q8N5K1 1/20 0.39
GAK O14976 1/20 0.38
RIPK2 O43353 1/20 0.38
STK16 O75716 1/20 0.38
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10745539 0.88 CSNK1D (0.41) ICAM1SELEVCAM1NPSR1CSNK1D
SCHEMBL10741832 0.86 CFTR (0.46) ICAM1SELEVCAM1MAPK1NPSR1
SCHEMBL8442991 0.81 ICAM1 (0.77) ICAM1SELEVCAM1PRNPTSHR
SCHEMBL9857130 0.80 ICAM1 (0.41) ICAM1SELEVCAM1DYRK1AKDM4E
SCHEMBL9857920 0.77 SENP5 (0.38) ICAM1SELEVCAM1HTTGAK
SCHEMBL693963 0.77 CYP2C19 (0.41) PRNPTSHRMAPK1PPARGHTT
SCHEMBL692750 0.76 CSNK1D (0.41) PRNPTSHRMAPK1PPARGHTT
SCHEMBL15697523 0.76 ALDH1A1 (0.59) MAPK1HTTNPSR1CFTRCISD2
SCHEMBL693546 0.76 ALDH1A1 (0.47) MAPK1MAPK10NPSR1CSNK1DCFTR
SCHEMBL15698889 0.75 CFTR (0.43) MAPK1MAPK10NPSR1CSNK1DCFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068248-A Analgesics, antipyretics and antiinflammatory agents MERCK & CO., INC. (US) 1991-11-26 US disclosed
EP-0160408-B1 BENZOTHIOPHENES, THEIR PRODUCTION AND USE, AND COMPOSITIONS CONTAINING THEM MERCK & CO. INC. (US) 1989-08-23 EP disclosed
US-4760086-A N-alkenyl-3-hydroxybenzo[b]thiophene-2-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-07-26 US disclosed
EP-0160408-A1 Benzothiophenes, their production and use, and compositions containing them MERCK & CO. INC. (US) 1985-11-06 EP disclosed