SCHEMBL9858313

SCHEMBL9858313

NC(=O)c1cn(Cc2cc(F)ccc2F)nn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA5A P35218 1/20 0.61
SCD O00767 1/20 0.51
GRM2 Q14416 3/20 0.46
TUBB4A P04350 2/20 0.45
TUBB P07437 2/20 0.45
TUBA3C P0DPH7 2/20 0.45
TUBA1B P68363 2/20 0.45
TUBA4A P68366 2/20 0.45
TUBB4B P68371 2/20 0.45
TUBB3 Q13509 2/20 0.45
TUBB2A Q13885 2/20 0.45
TUBB8 Q3ZCM7 2/20 0.45
TUBA3E Q6PEY2 2/20 0.45
TUBA1A Q71U36 2/20 0.45
TUBA1C Q9BQE3 2/20 0.45
TUBB6 Q9BUF5 2/20 0.45
TUBB2B Q9BVA1 2/20 0.45
TUBB1 Q9H4B7 2/20 0.45
RIPK1 Q13546 1/20 0.43
HDAC1 Q13547 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857419 0.89 CA5A (0.61) CA5ASCDGRM2HDAC1USP2
SCHEMBL30645406 0.83 CA5A (0.72) CA5ASCDHDAC1ALDH1A1MAPT
SCHEMBL9857405 0.83 CA5A (0.72) CA5ASCDHDAC1ALDH1A1MAPT
SCHEMBL17283081 0.83 TUBB4A (0.47) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL20344482 0.80 CA5A (0.63) CA5ASCDGRM2TUBB4ATUBB
SCHEMBL9857834 0.78 CA5A (0.73) CA5ASCDGRM2HDAC1ALDH1A1
SCHEMBL15964868 0.78 CA5A (0.65) CA5ASCDGRM2TUBB4ATUBB
Rufinamide SCHEMBL230448 0.76 CA5A (1.00) CA5ASCDGRM2ALDH1A1KLKB1
Rufinamide SCHEMBL20769779 0.76 CA5A (1.00) CA5ASCDGRM2ALDH1A1KLKB1
SCHEMBL9714457 0.76 GRM2 (0.43) CA5AGRM2RIPK1DPP4MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP disclosed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US disclosed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP disclosed