SCHEMBL9860146

SCHEMBL9860146

CC1(C)CC(=O)C(C)(C)c2ccc(Br)cc21

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 1/20 0.40
AHR P35869 1/20 0.40
TDP2 O95551 1/20 0.38
PDE4B Q07343 1/20 0.36
ALDH1A1 P00352 3/20 0.35
BACE1 P56817 4/20 0.35
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NR2F2 P24468 1/20 0.33
HSD17B10 Q99714 1/20 0.33
BRD4 O60885 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9860639 0.93 CMA1 (0.40) CMA1AHRTDP2PDE4BALDH1A1
SCHEMBL9418964 0.81 CMA1 (0.42) CMA1AHRTDP2PDE4BALDH1A1
SCHEMBL13716890 0.80 PGR (0.40) ALDH1A1MAPTKMT2AKDM4EHPGD
SCHEMBL10452858 0.75 PDK2 (0.41) ALDH1A1KMT2ANR2F2KDM4EHPGD
SCHEMBL8511471 0.75 CYP26A1 (0.41) CMA1AHRTDP2ALDH1A1KMT2A
SCHEMBL10453208 0.75 RARB (0.43) ALDH1A1TP53MAPTKMT2ASMN1; SMN2
SCHEMBL25244202 0.74 RXRA (0.37)
SCHEMBL12721438 0.74 CYP2A6 (0.35) CMA1AHRALDH1A1
SCHEMBL20212018 0.74 CYP2A6 (0.35) CMA1AHRALDH1A1
SCHEMBL13717001 0.74 BCHE (0.38) ALDH1A1BACE1KMT2AKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5055622-A For treating neoplasms and dermatoses HOFFMANN-LA ROCHE INC. (US) 1991-10-08 US disclosed
US-5030764-A Antitumor agents; treatment of skin disorders HOFFMANN-LA ROCHE INC. (US) 1991-07-09 US disclosed
US-5030765-A Skin disorders, anititumor agents HOFFMANN-LA ROCHE INC. (US) 1991-07-09 US disclosed
US-5001276-A Novel tetrahydronaphthalene and indane derivatives HOFFMANN-LA ROCHE INC. (US) 1991-03-19 US disclosed
US-4990703-A Novel tetrahydronaphthalene and indane derivatives HOFFMANN-LA ROCHE INC. (US) 1991-02-05 US disclosed
US-4935560-A ANTITUMOR AGENTS; SKIN DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-06-19 US disclosed
US-4870219-A NEOPLASMS, DERMATOSES HOFFMANN-LA ROCHE INC. (US) 1989-09-26 US disclosed