SCHEMBL9860258

SCHEMBL9860258

CC(I)C(N)(N)Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.56
SLC6A2 P23975 3/20 0.56
TRPA1 O75762 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
HIF1A Q16665 1/20 0.45
SIGMAR1 Q99720 2/20 0.45
MAOA P21397 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
CYP2A6 P11509 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
CYP2D6 P10635 2/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
EPHX1 P07099 1/20 0.38
CYP3A4 P08684 1/20 0.38
RECQL P46063 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8761557 0.81 SLC6A2 (0.54) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A
SCHEMBL8915534 0.79 TAAR1 (0.52) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A
SCHEMBL18886612 0.76 TAAR1 (0.58) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A
SCHEMBL18426836 0.74 SLC6A2 (0.56) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A
SCHEMBL10508831 0.74 TAAR1 (0.56) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A
SCHEMBL3663463 0.74 SLC6A2 (0.56) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A
SCHEMBL10503241 0.73 TAAR1 (0.67) TAAR1SLC6A2SMN1; SMN2HIF1AMAOA
SCHEMBL2487465 0.72 TAAR1 (0.73) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A
Phentermine SCHEMBL26615 0.72 SLC6A2 (1.00) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A
SCHEMBL22304553 0.72 SLC6A2 (0.58) TAAR1SLC6A2TRPA1SMN1; SMN2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021220-A Haluaromatic compound, water-soluble acid, copper salt acid-stable reducing agent MALLINCKRODT, INC. (US) 1991-06-04 US disclosed
US-4942231-A CATALYTIC HALOGENATION IN THE PRESENCE OF A REDUCING AGENT AND ACID MEDIUM MALLINCKRODT, INC. (US) 1990-07-17 US disclosed
EP-0165630-B1 METHOD OF PREPARING A CHLORINATED, BROMINATED, RADIOBROMINATED, IODINATED AND/OR RADIOIODINATED, AROMATIC OR HETEROAROMATIC COMPOUND, AS WELL AS A KIT FOR PREPARING A DIAGNOSTIC COMPOSITION ON THE BASIS OF THIS COMPOUND MALLINCKRODT, INC.(a Missouri corporation) (US) 1989-10-18 EP disclosed
EP-0165630-A2 Method of preparing a chlorinated, brominated, radiobrominated, iodinated and/or radioiodinated, aromatic or heteroaromatic compound, as well as a kit for preparing a diagnostic composition on the basis of this compound MALLINCKRODT, INC.(a Missouri corporation) (US) 1985-12-27 EP disclosed