SCHEMBL9860426

SCHEMBL9860426

CCOS(=O)(=O)C(CC)c1ccccc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
PSIP1 O75475 1/20 0.37
CYP3A4 P08684 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MC4R P32245 3/20 0.35
KCNQ2 O43526 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
IDO1 P14902 2/20 0.33
TDO2 P48775 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CES2 O00748 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31111607 0.78 CA12 (0.41) CA12CA1CA2CA9PSIP1
SCHEMBL27540936 0.78 PSIP1 (0.40) CA12CA1CA2CA9PSIP1
Hydrochloric Acid SCHEMBL31111474 0.77 CA12 (0.40) CA12CA1CA2CA9PSIP1
SCHEMBL3884592 0.75 PSIP1 (0.40) CA12CA1CA2CA9PSIP1
SCHEMBL779565 0.73 CA12 (0.43) CA12CA1CA2CA9PSIP1
SCHEMBL3883384 0.72 CYP3A4 (0.40) CA12CA1CA2CA9PSIP1
SCHEMBL781961 0.70 TSHR (0.40) PSIP1CYP3A4L3MBTL1MC4RKCNQ2
SCHEMBL15431689 0.69 PSIP1 (0.38) CA12CA1CA2CA9PSIP1
SCHEMBL7984628 0.69 IDO1 (0.40) CA12CA1CA2CA9PSIP1
SCHEMBL15431686 0.69 PSIP1 (0.38) CA12CA1CA2CA9PSIP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5055622-A For treating neoplasms and dermatoses HOFFMANN-LA ROCHE INC. (US) 1991-10-08 US disclosed
US-5030765-A Skin disorders, anititumor agents HOFFMANN-LA ROCHE INC. (US) 1991-07-09 US disclosed
US-5030764-A Antitumor agents; treatment of skin disorders HOFFMANN-LA ROCHE INC. (US) 1991-07-09 US disclosed
US-5001276-A Novel tetrahydronaphthalene and indane derivatives HOFFMANN-LA ROCHE INC. (US) 1991-03-19 US disclosed
US-4990703-A Novel tetrahydronaphthalene and indane derivatives HOFFMANN-LA ROCHE INC. (US) 1991-02-05 US disclosed
US-4935560-A ANTITUMOR AGENTS; SKIN DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-06-19 US disclosed
US-4870219-A NEOPLASMS, DERMATOSES HOFFMANN-LA ROCHE INC. (US) 1989-09-26 US disclosed