SCHEMBL9860748

SCHEMBL9860748

Brc1cc2ncccc2c2ncccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.59
HTT P42858 5/20 0.59
HSP90AA1 P07900 4/20 0.59
TDP1 Q9NUW8 3/20 0.59
TP53 P04637 3/20 0.59
SMN1; SMN2 Q16637 3/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
USP2 O75604 1/20 0.59
LMNA P02545 3/20 0.55
MAPT P10636 4/20 0.50
ALDH1A1 P00352 3/20 0.50
APAF1 O14727 1/20 0.50
TDP2 O95551 1/20 0.50
CASP3 P42574 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
L3MBTL1 Q9Y468 3/20 0.42
NPC1 O15118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9976765 0.85 KDM4E (0.66) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL22117512 0.82 MAPT (0.54) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL27934157 0.78 MEN1 (0.58) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL22117517 0.78 KDM4E (0.58) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL18935217 0.78 KDM4E (0.49) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL3711428 0.78 KDM4E (0.45) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL29551392 0.78 HTT (0.52) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL4470656 0.78 HTT (0.52) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL1149641 0.76 L3MBTL1 (0.61) KDM4EHTTHSP90AA1TDP1TP53
SCHEMBL8654916 0.76 CCR1 (0.61) KDM4EHTTHSP90AA1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110818739-B Metal iridium complex with synergistic response to tumor microenvironment pH/hypoxic and application thereof 南京大学 2021-05-28 CN disclosed
CN-110857310-B Polyamphidine ruthenium complex with photoactivity and application thereof 南京大学 2021-05-28 CN disclosed
CN-110857310-A Polyamphidine ruthenium complex with photoactivity and application thereof 南京大学 2020-03-03 CN disclosed
CN-110818739-A Metal iridium complex with synergistic response to tumor microenvironment pH/hypoxic and application thereof 南京大学 2020-02-21 CN disclosed
US-5070158-A Covalently labeled siloxane polymers HEWLETT-PACKARD COMPANY (US) 1991-12-03 US disclosed
EP-0283206-A2 Covalently labeled siloxane polymers Hewlett-Packard Company (US) 1988-09-21 EP disclosed