SCHEMBL9861314

SCHEMBL9861314

CCc1cc(C(F)(F)C(F)(F)C(F)(F)F)ccc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
ALDH1A1 P00352 2/20 0.39
POLB P06746 2/20 0.39
ESR1 P03372 5/20 0.36
ESR2 Q92731 4/20 0.36
AR P10275 2/20 0.34
FFAR4 Q5NUL3 2/20 0.33
KIF11 P52732 1/20 0.33
LMNA P02545 2/20 0.32
FFAR1 O14842 1/20 0.31
ATM Q13315 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CFTR P13569 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PGR P06401 1/20 0.31
HSD11B1 P28845 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6690284 0.89 MAPT (0.41) MAPTALDH1A1POLBESR1ESR2
SCHEMBL5958735 0.82 MAPT (0.45) MAPTALDH1A1POLBESR1ESR2
SCHEMBL8369193 0.82 ALDH1A1 (0.46) MAPTALDH1A1POLBESR1ESR2
SCHEMBL5958646 0.80 HTT (0.40) MAPTALDH1A1POLBESR1ESR2
SCHEMBL7096170 0.79 NR1H2 (0.47) LMNASMN1; SMN2HSD17B10PGR
SCHEMBL9861430 0.79 ESR1 (0.61) ESR1ESR2AR
SCHEMBL3910479 0.78 CYP3A4 (0.45) MAPTALDH1A1ESR1ESR2AR
SCHEMBL5230955 0.78 MAPT (0.38) MAPTALDH1A1POLBESR1ESR2
SCHEMBL16150691 0.77 MAPT (0.37) MAPTALDH1A1POLBESR1ESR2
SCHEMBL5958760 0.77 KLF10 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed