SCHEMBL9861385

SCHEMBL9861385

Nc1c(C2CCCC2)cc(C(F)(F)F)c2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
BACE1 P56817 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GAA P10253 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALOX5AP P20292 3/20 0.35
FEN1 P39748 3/20 0.35
CAMKK2 Q96RR4 1/20 0.35
RBP4 P02753 2/20 0.35
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9862064 0.81 GAA (0.41) HTR2CBACE1KDM4EMEN1MAPT
SCHEMBL9861402 0.73 HTR2C (0.49) HTR2CGAATDP1ALOX5APFEN1
SCHEMBL29721046 0.72 HTR2C (0.70) HTR2CGAATDP1RBP4CUL4A
SCHEMBL1919230 0.72 HTR2C (0.70) HTR2CGAATDP1RBP4CUL4A
SCHEMBL29720917 0.71 HTR2C (0.68) HTR2CGAATDP1RBP4CUL4A
SCHEMBL15156609 0.71 HTR2C (0.68) HTR2CGAATDP1RBP4CUL4A
SCHEMBL13349962 0.70 TSHR (0.50) HTR2CMAPK1GAA
SCHEMBL24332883 0.69 KDM4E (0.47) LMNASMN1; SMN2BACE1KDM4EMEN1
SCHEMBL9861395 0.69 KMT2A (0.47) LMNASMN1; SMN2BACE1KDM4EMEN1
SCHEMBL28247607 0.69 HTR2C (0.70) HTR2CGAATDP1RBP4CUL4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed