SCHEMBL9861395

SCHEMBL9861395

Cc1cc(C(F)(F)F)c2ccccc2c1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.47
MEN1 O00255 4/20 0.47
KDM4E B2RXH2 3/20 0.47
BACE1 P56817 2/20 0.47
MAPT P10636 2/20 0.47
LMNA P02545 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PARP1 P09874 1/20 0.38
AR P10275 3/20 0.38
EP300 Q09472 1/20 0.37
PKM P14618 1/20 0.36
HSD11B1 P28845 1/20 0.35
POLB P06746 3/20 0.35
GLA P06280 2/20 0.35
GAA P10253 2/20 0.35
TSHR P16473 2/20 0.35
PTPN1 P18031 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861512 0.85 KDM4E (0.53) KMT2AMEN1KDM4EBACE1MAPT
SCHEMBL11412130 0.82 MEN1 (0.73) KMT2AMEN1KDM4EMAPTLMNA
SCHEMBL11412134 0.82 KDM4E (0.54) KMT2AMEN1KDM4EBACE1MAPT
SCHEMBL9861634 0.79 KDM4E (0.54) KMT2AMEN1KDM4EBACE1MAPT
SCHEMBL24332883 0.77 KDM4E (0.47) KMT2AMEN1KDM4EBACE1MAPT
SCHEMBL9861488 0.77 HTT (0.57) KMT2AMEN1KDM4EBACE1MAPT
SCHEMBL9861455 0.77 KDM4E (0.44) KMT2AMEN1KDM4EBACE1MAPT
SCHEMBL9861337 0.77 KDM4E (0.44) KMT2AMEN1KDM4EBACE1MAPT
SCHEMBL1562090 0.74 CYP1A2 (0.50) KDM4EBACE1LMNASMN1; SMN2EP300
SCHEMBL29462977 0.74 CYP1A2 (0.43) KDM4EBACE1LMNAHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed