SCHEMBL9861337

SCHEMBL9861337

CC(C)c1cc(C(F)(F)F)c2ccccc2c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
MAPT P10636 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
BACE1 P56817 1/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
AR P10275 4/20 0.36
TRPA1 O75762 1/20 0.36
EP300 Q09472 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
P2RX7 Q99572 1/20 0.33
GAA P10253 3/20 0.33
ALDH1A1 P00352 3/20 0.33
GLA P06280 2/20 0.33
POLB P06746 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861417 0.87 KDM4E (0.49) KDM4EKMT2AMEN1MAPTNPSR1
SCHEMBL9861997 0.79 BCL2 (0.41) BACE1LMNAHTTARTRPA1
SCHEMBL9861508 0.77 KCNH2 (0.36) KDM4EKMT2AMEN1MAPTNPSR1
SCHEMBL9861395 0.77 KMT2A (0.47) KDM4EKMT2AMEN1MAPTNPSR1
SCHEMBL9861634 0.75 KDM4E (0.54) KDM4EKMT2AMEN1MAPTNPSR1
SCHEMBL24910099 0.74 P2RX7 (0.37) BACE1SMN1; SMN2ARTRPA1NR1H2
SCHEMBL28883418 0.73 CYP1A2 (0.39) KDM4EKMT2AMEN1MAPTLMNA
SCHEMBL24332883 0.73 KDM4E (0.47) KDM4EKMT2AMEN1MAPTNPSR1
SCHEMBL9861455 0.72 KDM4E (0.44) KDM4EKMT2AMEN1MAPTNPSR1
SCHEMBL9861638 0.71 P2RX7 (0.49) LMNAARTRPA1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed