SCHEMBL9861455

SCHEMBL9861455

CCc1cc(C(F)(F)F)c2ccccc2c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
HTT P42858 2/20 0.44
BACE1 P56817 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
AR P10275 9/20 0.43
TRPA1 O75762 1/20 0.36
IDO1 P14902 2/20 0.36
PTGES O14684 1/20 0.34
EP300 Q09472 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
SRC P12931 1/20 0.34
HPGD P15428 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861499 0.84 KDM4E (0.46) KDM4EMEN1KMT2ANPSR1HTT
SCHEMBL9861341 0.80 BACE1 (0.45) KDM4EMEN1KMT2ANPSR1HTT
SCHEMBL9861301 0.79 GABRA1 (0.44) BACE1ARTRPA1
SCHEMBL9861395 0.77 KMT2A (0.47) KDM4EMEN1KMT2ANPSR1HTT
SCHEMBL9778555 0.76 PKM (0.42) KDM4EMEN1KMT2ANPSR1HTT
SCHEMBL9861634 0.75 KDM4E (0.54) KDM4EMEN1KMT2ANPSR1HTT
SCHEMBL24332883 0.73 KDM4E (0.47) KDM4EMEN1KMT2ANPSR1HTT
SCHEMBL28883537 0.73 CYP1A2 (0.39) KDM4EMEN1KMT2AHTTLMNA
SCHEMBL9861337 0.72 KDM4E (0.44) KDM4EMEN1KMT2ANPSR1HTT
SCHEMBL9861905 0.71 GABRA1 (0.45) KMT2ANPSR1LMNAMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed