SCHEMBL9861418

SCHEMBL9861418

O=C1C=CC(O)(C(F)(F)F)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 19/20 0.48
IDO1 P14902 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
CDC25B P30305 1/20 0.43
AKT1 P31749 1/20 0.43
SNCA P37840 1/20 0.43
MAP2K1 Q02750 1/20 0.43
PIN1 Q13526 1/20 0.43
EHMT2 Q96KQ7 1/20 0.43
NSD1 Q96L73 1/20 0.43
EHMT1 Q9H9B1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6917185 0.76 IDO1 (0.52) PDK2IDO1MAOAMAOBCDC25B
SCHEMBL9861969 0.70 PDK2 (0.46) PDK2
SCHEMBL13508801 0.69 CDC25B (0.43) IDO1MAOAMAOBCDC25BAKT1
SCHEMBL30229349 0.68 IDO1 (0.46) PDK2IDO1MAOAMAOBCDC25B
SCHEMBL9861622 0.68 PDK2 (0.76) PDK2
Naphthoquinone SCHEMBL28997832 0.66 IDO1 (0.70) PDK2IDO1MAOAMAOBCDC25B
SCHEMBL15463143 0.66 PDK2 (1.00) PDK2
SCHEMBL9861348 0.66 PDK2 (0.35) PDK2
Naphthoquinone SCHEMBL28297132 0.66 CDC25B (0.78) IDO1MAOAMAOBCDC25BAKT1
SCHEMBL10554281 0.66 PDK2 (0.53) PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed