SCHEMBL9861532

SCHEMBL9861532

CCc1cc(C(F)(F)C(F)(F)F)ccc1O

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.65
ESR2 Q92731 6/20 0.65
KLF10 Q13118 1/20 0.46
BACE1 P56817 1/20 0.43
CYP2D6 P10635 2/20 0.42
HSD17B1 P14061 2/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
AR P10275 2/20 0.40
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
CACNA1B Q00975 1/20 0.37
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861430 0.89 ESR1 (0.61) ESR1ESR2KLF10BACE1CYP2D6
SCHEMBL20958252 0.85 ESR1 (0.65) ESR1ESR2KLF10BACE1CYP2D6
SCHEMBL178283 0.85 ESR1 (0.69) ESR1ESR2KLF10BACE1CYP2D6
SCHEMBL28738556 0.80 ESR1 (0.57) ESR1ESR2KLF10BACE1CYP2D6
SCHEMBL122862 0.79 ESR1 (0.71) ESR1ESR2KLF10BACE1CYP2D6
SCHEMBL1229448 0.79 ESR1 (0.71) ESR1ESR2KLF10BACE1CYP2D6
SCHEMBL8062965 0.79 ESR1 (0.71) ESR1ESR2KLF10BACE1CYP2D6
SCHEMBL29395018 0.79 ESR1 (0.71) ESR1ESR2KLF10BACE1CYP2D6
SCHEMBL9861336 0.79 GABRA1 (0.46) ESR1ESR2ARGABRA1GABRB2
SCHEMBL30234175 0.79 ESR1 (0.71) ESR1ESR2KLF10BACE1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed