SCHEMBL9861981

SCHEMBL9861981

COCc1ccccc1CNC(C)=O

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SETDB1 Q15047 1/20 0.49
MTNR1A P48039 4/20 0.49
MTNR1B P49286 3/20 0.49
NPSR1 Q6W5P4 2/20 0.44
CACNA1G O43497 1/20 0.44
CACNA1H O95180 1/20 0.44
CACNA1I Q9P0X4 1/20 0.44
HPGD P15428 2/20 0.44
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
HTT P42858 1/20 0.42
ALDH1A1 P00352 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
NQO2 P16083 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14204990 0.87 SETDB1 (0.59) SETDB1MTNR1AMTNR1BNPSR1HPGD
SCHEMBL3918538 0.86 HPGD (0.47) NPSR1CACNA1GCACNA1HCACNA1IHPGD
SCHEMBL15716617 0.84 NPSR1 (0.44) MTNR1AMTNR1BNPSR1CACNA1GCACNA1H
SCHEMBL14651452 0.81 SETDB1 (0.54) SETDB1MTNR1AMTNR1BNPSR1HPGD
SCHEMBL14651456 0.80 SETDB1 (0.44) SETDB1MTNR1AMTNR1BNPSR1HPGD
SCHEMBL29675775 0.79 SETDB1 (0.53) SETDB1MTNR1AMTNR1BNPSR1HPGD
SCHEMBL31531439 0.79 KMT2A (0.45) NPSR1CACNA1GCACNA1HCACNA1IHPGD
SCHEMBL10781979 0.79 SETDB1 (0.49) SETDB1MTNR1AMTNR1BNPSR1HPGD
SCHEMBL885000 0.79 MTNR1A (0.71) MTNR1AMTNR1BNPSR1HPGDKMT2A
SCHEMBL1799028 0.78 SETDB1 (0.51) SETDB1MTNR1AMTNR1BNPSR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108617166-B Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-05-17 CN claimed
US-4992588-A Preparation of o-acylaminomethylbenzyl halides BASF AKTIENGESELLSCHAFT (DE) 1991-02-12 US disclosed
EP-0087676-B1 PROCESS FOR THE PREPARATION OF O-ACYLAMINOMETHYLBENZYL HALOGENIDES BASF Aktiengesellschaft (DE) 1987-12-16 EP disclosed
EP-0087676-A1 Process for the preparation of o-acylaminomethylbenzyl halogenides BASF Aktiengesellschaft (DE) 1983-09-07 EP disclosed