SCHEMBL9864052

SCHEMBL9864052

CC(C)(CC(N)C1(c2ccc(Cl)cc2)CCC1)OC(=O)/C=C\C(=O)OC(C)(C)CC(N)C1(c2ccc(Cl)cc2)CCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.50
SLC6A3 Q01959 11/20 0.50
CYP3A4 P08684 4/20 0.50
ALOX15 P16050 2/20 0.50
TSHR P16473 2/20 0.50
TP53 P04637 1/20 0.50
SLC6A2 P23975 5/20 0.41
CHRM2 P08172 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
HTR2A P28223 1/20 0.38
OPRK1 P41145 1/20 0.38
HTR2B P41595 1/20 0.38
KCNH2 Q12809 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
NFKB1 P19838 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9864002 0.88 SLC6A4 (0.50) SLC6A4SLC6A3CYP3A4ALOX15TSHR
SCHEMBL9864026 0.84 SLC6A3 (0.53) SLC6A4SLC6A3CYP3A4ALOX15TSHR
Fumaric Acid SCHEMBL9864056 0.80 SLC6A4 (0.51) SLC6A4SLC6A3CYP3A4ALOX15TSHR
Maleic Acid SCHEMBL9864047 0.80 SLC6A4 (0.51) SLC6A4SLC6A3CYP3A4ALOX15TSHR
SCHEMBL5661116 0.79 SLC6A4 (0.61) SLC6A4SLC6A3CYP3A4ALOX15TSHR
SCHEMBL7049796 0.79 SLC6A4 (0.61) SLC6A4SLC6A3CYP3A4ALOX15TSHR
SCHEMBL5668946 0.79 SLC6A4 (0.61) SLC6A4SLC6A3CYP3A4ALOX15TSHR
Maleic Acid SCHEMBL9863998 0.77 SLC6A4 (0.51) SLC6A4SLC6A3CYP3A4ALOX15TSHR
Fumaric Acid SCHEMBL9864009 0.77 SLC6A4 (0.51) SLC6A4SLC6A3CYP3A4ALOX15TSHR
SCHEMBL9864319 0.76 SLC6A4 (0.58) SLC6A4SLC6A3CYP3A4ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047432-A Antidepressants THE BOOTS COMPANY PLC (GB) 1991-09-10 US disclosed
US-4925879-A ANTIDEPRESSANTS BOOTS COMPANY, PLC (GB) 1990-05-15 US disclosed
EP-0191542-B1 ARYLCYCLOBUTYLALKYL AMINES AND THEIR USE AS ANTIDEPRESSIVE MEDICINES The Boots Company PLC (GB) 1988-06-08 EP disclosed