SCHEMBL9864070

SCHEMBL9864070

O=c1c(CCCl)n[nH]c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.53
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 4/20 0.50
RAB9A P51151 4/20 0.50
NPC1 O15118 3/20 0.50
TP53 P04637 1/20 0.50
GAA P10253 4/20 0.43
PDPK1 O15530 1/20 0.43
CYP3A4 P08684 1/20 0.43
HPGD P15428 2/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GLA P06280 1/20 0.41
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.41
CTNNB1 P35222 1/20 0.41
WNT3A P56704 1/20 0.41
IDO1 P14902 2/20 0.41
ALPL P05186 1/20 0.41
TTK P33981 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23908909 0.83 CYP1A2 (0.53) CYP1A2KDM4EALDH1A1RAB9ANPC1
SCHEMBL30727481 0.83 CYP1A2 (0.53) CYP1A2KDM4EALDH1A1RAB9ANPC1
SCHEMBL21591507 0.81 CYP1A2 (0.58) CYP1A2KDM4EALDH1A1RAB9ANPC1
SCHEMBL9078088 0.80 CYP1A2 (0.49) CYP1A2KDM4EALDH1A1RAB9ANPC1
SCHEMBL11806745 0.80 CTNNB1 (0.51) CYP1A2KDM4EALDH1A1RAB9ANPC1
SCHEMBL9865079 0.76 AR (0.44) CYP1A2KDM4ERAB9AHPGDLMNA
SCHEMBL320109 0.76 KDM4E (0.46) CYP1A2KDM4EALDH1A1RAB9ANPC1
SCHEMBL23908935 0.75 LMNA (0.62) CYP1A2KDM4EALDH1A1RAB9ANPC1
SCHEMBL960151 0.74 KDM4E (0.52) CYP1A2KDM4EALDH1A1RAB9ANPC1
SCHEMBL23909017 0.71 SMN1; SMN2 (0.66) CYP1A2KDM4EALDH1A1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988695-A Gastrointestinal disorders, antisecretory agents SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-01-29 US disclosed
EP-0380257-A2 Condensed cinnoline derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them SMITHKLINE BECKMAN INTERCREDIT B.V. (NL) 1990-08-01 EP disclosed