SCHEMBL98641

SCHEMBL98641

CCc1nc(SCc2ccc(OC)c(C#N)c2)nc2c1nc(N)n2C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.39
ALDH1A1 P00352 6/20 0.38
KDM4E B2RXH2 5/20 0.38
KMT2A Q03164 3/20 0.38
HSD17B10 Q99714 3/20 0.38
HPGD P15428 2/20 0.38
GAA P10253 2/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
USP2 O75604 2/20 0.37
MAOB P27338 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
AR P10275 2/20 0.35
MEN1 O00255 2/20 0.34
CNR2 P34972 1/20 0.34
GLA P06280 1/20 0.33
DCUN1D1 Q96GG9 4/20 0.33
UBE2M P61081 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL97698 0.87 GAA (0.39) ALDH1A1KMT2AGAAMAPTL3MBTL1
SCHEMBL98718 0.78 GSK3B (0.36) GSK3BALDH1A1GAAMAOBL3MBTL1
SCHEMBL171495 0.74 KDM1A (0.34) GSK3BALDH1A1KDM4EKMT2AHPGD
SCHEMBL97922 0.74 PIK3CA (0.43) GSK3BALDH1A1KDM4EHSD17B10HPGD
SCHEMBL97709 0.73 CCNE2 (0.41) GSK3BCASP1MAOB
SCHEMBL98983 0.72 GSK3B (0.36) GSK3BALDH1A1MAPTMAOBL3MBTL1
SCHEMBL98560 0.72 GSK3B (0.37) GSK3BALDH1A1GAAMAPTMAOB
SCHEMBL98972 0.72 YTHDC1 (0.41) GSK3BMAOB
SCHEMBL99189 0.72 GSK3B (0.38) GSK3BALDH1A1HSD17B10HPGDMAOB
SCHEMBL98435 0.69 CSF1R (0.41) GSK3BALDH1A1KDM4EHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426130-B1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KK (JP) 2015-03-11 EP disclosed
EP-2426130-A1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 2012-03-07 EP disclosed