SCHEMBL9864157

SCHEMBL9864157

CSCCCC(N(C)C)C1(c2ccc(Cl)c(Cl)c2)CCC1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 16/20 0.62
SLC6A4 P31645 16/20 0.62
SLC6A2 P23975 12/20 0.52
KCNH2 Q12809 5/20 0.52
CHRM2 P08172 1/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
HTR2A P28223 1/20 0.45
OPRK1 P41145 1/20 0.45
HTR2B P41595 1/20 0.45
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9864283 0.86 SLC6A3 (0.61) SLC6A3SLC6A4SLC6A2KCNH2CHRM2
SCHEMBL9864143 0.85 SLC6A3 (0.64) SLC6A3SLC6A4SLC6A2KCNH2CHRM2
SCHEMBL6392408 0.85 SLC6A3 (0.64) SLC6A3SLC6A4SLC6A2KCNH2CHRM2
SCHEMBL10543400 0.83 SLC6A3 (0.73) SLC6A3SLC6A4SLC6A2KCNH2CHRM2
SCHEMBL9864037 0.83 SLC6A3 (0.62) SLC6A3SLC6A4SLC6A2KCNH2CHRM2
SCHEMBL9864378 0.83 SLC6A3 (0.62) SLC6A3SLC6A4SLC6A2KCNH2CHRM2
SCHEMBL9864406 0.82 SLC6A4 (0.69) SLC6A3SLC6A4SLC6A2KCNH2CYP3A4
Hydrochloric Acid SCHEMBL2729 0.82 SLC6A3 (0.71) SLC6A3SLC6A4SLC6A2KCNH2CHRM2
SCHEMBL31107082 0.82 SLC6A3 (0.72) SLC6A3SLC6A4SLC6A2KCNH2CHRM2
SCHEMBL31107083 0.82 SLC6A3 (0.72) SLC6A3SLC6A4SLC6A2KCNH2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047432-A Antidepressants THE BOOTS COMPANY PLC (GB) 1991-09-10 US disclosed
US-4925879-A ANTIDEPRESSANTS BOOTS COMPANY, PLC (GB) 1990-05-15 US disclosed
EP-0191542-B1 ARYLCYCLOBUTYLALKYL AMINES AND THEIR USE AS ANTIDEPRESSIVE MEDICINES The Boots Company PLC (GB) 1988-06-08 EP disclosed
EP-0191542-A1 Arylcyclobutylalkyl amines and their use as antidepressive medicines The Boots Company PLC (GB) 1986-08-20 EP disclosed