SCHEMBL9864259

SCHEMBL9864259

CCC(=O)C(N(C)CCN1CCOCC1)C1(c2ccc(Cl)c(Cl)c2)CCC1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45
SLC6A3 Q01959 10/20 0.43
SLC6A4 P31645 9/20 0.43
SLC6A2 P23975 7/20 0.43
TACR3 P29371 1/20 0.42
SIGMAR1 Q99720 4/20 0.41
KCNH2 Q12809 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9864574 0.83 SLC6A3 (0.49) SLC6A3SLC6A4SLC6A2KCNH2
SCHEMBL9864332 0.82 CASR (0.44) TACR3
SCHEMBL10839380 0.81 CHRM2 (0.48) CHRM2CHRM1SLC6A3SLC6A4SLC6A2
SCHEMBL9864123 0.79 SLC6A3 (0.57) SLC6A3SLC6A4SLC6A2KCNH2
Hydrochloric Acid SCHEMBL10839808 0.76 KCNH2 (0.48) CHRM2CHRM1SLC6A3SLC6A4SLC6A2
Hydrochloric Acid SCHEMBL10840534 0.76 KCNH2 (0.48) CHRM2CHRM1SLC6A3SLC6A4SLC6A2
SCHEMBL9863839 0.73 SLC6A3 (0.50) SLC6A3SLC6A4SLC6A2KCNH2
SCHEMBL9864639 0.72 SLC6A3 (0.50) SLC6A3SLC6A4SLC6A2KCNH2
Hydrochloric Acid SCHEMBL10839009 0.72 SLC6A2 (0.51) CHRM2CHRM1SLC6A3SLC6A4SLC6A2
SCHEMBL16523028 0.72 SLC6A4 (0.55) CHRM2CHRM1SLC6A3SLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047432-A Antidepressants THE BOOTS COMPANY PLC (GB) 1991-09-10 US disclosed
US-4925879-A ANTIDEPRESSANTS BOOTS COMPANY, PLC (GB) 1990-05-15 US disclosed
EP-0191542-A1 Arylcyclobutylalkyl amines and their use as antidepressive medicines The Boots Company PLC (GB) 1986-08-20 EP disclosed