SCHEMBL9864332

SCHEMBL9864332

CCC(=O)C(N(C)CCN1CCOCC1)C1(c2cccc(C(F)(F)F)c2)CCC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.44
OPRM1 P35372 5/20 0.43
OPRL1 P41146 3/20 0.43
TACR1 P25103 2/20 0.41
TACR3 P29371 2/20 0.41
KMT2A Q03164 1/20 0.41
EPHX2 P34913 1/20 0.39
OPRD1 P41143 2/20 0.39
KDM4E B2RXH2 3/20 0.39
TRPV4 Q9HBA0 3/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9864129 0.83 CASR (0.41) CASROPRM1OPRL1TACR1TACR3
SCHEMBL9864259 0.82 CHRM2 (0.45) TACR3
SCHEMBL9864288 0.81 SLC6A4 (0.47) OPRM1OPRL1
SCHEMBL10638666 0.79 TACR3 (0.33) CASROPRM1OPRL1TACR1TACR3
SCHEMBL9864273 0.73 SLC6A4 (0.46) OPRM1OPRL1ALDH1A1
SCHEMBL9864359 0.65 SLC6A4 (0.48) OPRM1OPRL1OPRD1
SCHEMBL9118387 0.65 SLC6A4 (0.52) OPRM1OPRL1
SCHEMBL9864574 0.64 SLC6A3 (0.49)
SCHEMBL9863909 0.64 SLC6A4 (0.46) OPRM1OPRL1OPRD1
SCHEMBL12125729 0.64 KMT2A (0.64) KMT2AEPHX2TRPV4ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047432-A Antidepressants THE BOOTS COMPANY PLC (GB) 1991-09-10 US disclosed
US-4925879-A ANTIDEPRESSANTS BOOTS COMPANY, PLC (GB) 1990-05-15 US disclosed
EP-0191542-A1 Arylcyclobutylalkyl amines and their use as antidepressive medicines The Boots Company PLC (GB) 1986-08-20 EP disclosed