SCHEMBL9864270

SCHEMBL9864270

CC(O)(CC(N)C1(c2ccc(F)cc2)CCC1)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
SLC6A3 Q01959 10/20 0.40
SLC6A4 P31645 10/20 0.40
NR1I2 O75469 4/20 0.38
RORC P51449 4/20 0.38
SLC6A2 P23975 5/20 0.37
TRPA1 O75762 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9863419 0.88 SLC6A4 (0.56) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL9863736 0.87 TP53 (0.43) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL9864286 0.84 SLC6A3 (0.43) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL9864477 0.82 SLC6A3 (0.44) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL9864713 0.82 SLC6A3 (0.42) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL9864312 0.79 TP53 (0.37) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL10900716 0.78 SLC6A3 (0.41) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL9864319 0.77 SLC6A4 (0.58) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL9864308 0.75 SLC6A3 (0.39) TP53CYP3A4ALOX15TSHRSLC6A3
SCHEMBL9864298 0.75 KDM4E (0.38) TP53CYP3A4ALOX15TSHRSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047432-A Antidepressants THE BOOTS COMPANY PLC (GB) 1991-09-10 US disclosed
US-4925879-A ANTIDEPRESSANTS BOOTS COMPANY, PLC (GB) 1990-05-15 US disclosed
EP-0191542-B1 ARYLCYCLOBUTYLALKYL AMINES AND THEIR USE AS ANTIDEPRESSIVE MEDICINES The Boots Company PLC (GB) 1988-06-08 EP disclosed
EP-0191542-A1 Arylcyclobutylalkyl amines and their use as antidepressive medicines The Boots Company PLC (GB) 1986-08-20 EP disclosed