SCHEMBL9864963

SCHEMBL9864963

C=CCN1C(C)=C(C(=O)OC)C(c2ccccc2C(F)(F)F)C2=C1COC2=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 3/20 0.42
CACNA1F O60840 1/20 0.42
CACNA1D Q01668 1/20 0.42
CACNA1S Q13698 1/20 0.42
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 5/20 0.41
HPGD P15428 5/20 0.41
GAA P10253 5/20 0.41
GLA P06280 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 5/20 0.40
CYP1A2 P05177 3/20 0.40
CYP3A4 P08684 3/20 0.40
ADORA3 P0DMS8 3/20 0.40
MAPT P10636 3/20 0.40
CYP2C9 P11712 3/20 0.40
CYP2C19 P33261 3/20 0.40
TSHR P16473 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9864858 0.89 ALDH1A1 (0.46) CACNA1CCACNA1FCACNA1DCACNA1SKDM4E
SCHEMBL10968855 0.87 CACNA1C (0.36) CACNA1CCACNA1FCACNA1DCACNA1SKDM4E
SCHEMBL11007467 0.81 ALDH1A1 (0.46) CACNA1CCACNA1FCACNA1DCACNA1SKDM4E
SCHEMBL11006171 0.80 KDM4E (0.45) CACNA1CCACNA1FCACNA1DCACNA1SKDM4E
SCHEMBL9557790 0.78 KDM4E (0.38) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL11004817 0.77 KDM4E (0.47) CACNA1CCACNA1FCACNA1DCACNA1SKDM4E
SCHEMBL10966704 0.76 KDM4E (0.39) CACNA1CCACNA1FCACNA1DCACNA1SKDM4E
SCHEMBL11008208 0.74 GPBAR1 (0.40) KDM4EALDH1A1GAAHTTCYP3A4
SCHEMBL8868882 0.73 KDM4E (0.39) CACNA1CCACNA1FCACNA1DCACNA1SKDM4E
SCHEMBL9865585 0.73 CYP1A2 (0.58) CACNA1CCACNA1FCACNA1DCACNA1SKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5026714-A Novel 1-alkyl-substituted 1,4-dihydropyridinelactone anti-diabetics BAYER AKTIENGESELLSCHAFT (DE) 1991-06-25 US disclosed