SCHEMBL9864858

SCHEMBL9864858

CCN1C(C)=C(C(=O)OC)C(c2ccccc2C(F)(F)F)C2=C1COC2=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
KDM4E B2RXH2 5/20 0.46
HPGD P15428 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
CACNA1C Q13936 3/20 0.44
CACNA1F O60840 1/20 0.44
CACNA1D Q01668 1/20 0.44
CACNA1S Q13698 1/20 0.44
GAA P10253 4/20 0.44
GLA P06280 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 4/20 0.43
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 3/20 0.43
ADORA3 P0DMS8 3/20 0.43
MAPT P10636 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
TSHR P16473 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11007467 0.92 ALDH1A1 (0.46) ALDH1A1KDM4ETDP1CACNA1CCACNA1F
SCHEMBL9557790 0.89 KDM4E (0.38) ALDH1A1KDM4EHPGDTDP1GAA
SCHEMBL9864963 0.89 CACNA1C (0.42) ALDH1A1KDM4EHPGDTDP1CACNA1C
SCHEMBL10966704 0.86 KDM4E (0.39) ALDH1A1KDM4EHPGDTDP1CACNA1C
SCHEMBL11006171 0.85 KDM4E (0.45) ALDH1A1KDM4EHPGDTDP1CACNA1C
SCHEMBL9689389 0.82 KDM4E (0.40) ALDH1A1KDM4ETDP1CACNA1CCACNA1F
SCHEMBL11004817 0.82 KDM4E (0.47) ALDH1A1KDM4EHPGDTDP1CACNA1C
SCHEMBL8868882 0.78 KDM4E (0.39) ALDH1A1KDM4ETDP1CACNA1CCACNA1F
SCHEMBL9867642 0.78 PYGL (0.46) ALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL9865516 0.77 PYGL (0.48) ALDH1A1KDM4ECACNA1CCACNA1FCACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5026714-A Novel 1-alkyl-substituted 1,4-dihydropyridinelactone anti-diabetics BAYER AKTIENGESELLSCHAFT (DE) 1991-06-25 US disclosed