SCHEMBL9865008

SCHEMBL9865008

CCNC1CC2CCC(C1)N2c1nc2c(cc1F)c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.53
CHRM2 P08172 1/20 0.53
DRD1 P21728 1/20 0.53
LMNA P02545 3/20 0.51
KDM4E B2RXH2 3/20 0.51
HSD17B10 Q99714 2/20 0.51
ABCC4 O15439 1/20 0.51
TOP2A P11388 3/20 0.46
TOP2B Q02880 3/20 0.46
CYP2C9 P11712 1/20 0.46
ATP6V1B2 P21281 1/20 0.46
TBXA2R P21731 1/20 0.46
EDNRA P25101 1/20 0.46
TARBP2 Q15633 1/20 0.46
ALDH1A1 P00352 2/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
DHFR P00374 1/20 0.45
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10654645 0.85 DPP4 (0.58) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9838624 0.84 DPP4 (0.62) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9838732 0.84 DPP4 (0.62) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9837344 0.84 DPP4 (0.62) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9865696 0.84 DPP4 (0.55) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9837356 0.82 DPP4 (0.60) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9865560 0.81 TOP2A (0.54) CHRM2LMNAKDM4EHSD17B10TOP2A
SCHEMBL9865549 0.81 KDM4E (0.63) LMNAKDM4EHSD17B10TOP2ATOP2B
SCHEMBL9837577 0.80 LMNA (0.58) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9150328 0.80 DPP4 (0.67) DPP4CHRM2DRD1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP claimed
US-4992546-A Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives WARNER-LAMBERT COMPANY (US) 1991-02-12 US disclosed
US-4968799-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1990-11-06 US disclosed
US-4962108-A A QUIN-4-ONE HAVING THE FOLLOWING RING SUBSTITUENTS; 1-ALKYL OR PHENYL, 3-CARBOXY DERIVATIVE, 6-FLUORO AND 8-BRIDGED N-HETEROCYCLIC RING WARNER-LAMBERT COMPANY (US) 1990-10-09 US disclosed
US-4923879-A CARBOXYLIC ACID DERIVATIVES WITH BRIDGED SIDECHAINS WARNER-LAMBERT COMPANY (US) 1990-05-08 US disclosed
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP disclosed