SCHEMBL9865225

SCHEMBL9865225

COC(=O)CCNC(=O)c1ccc(O)c(NC(=O)c2ccc(C(=N)NC(=O)OC(C)(C)C)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.47
F10 P00742 1/20 0.40
PRSS1 P07477 1/20 0.40
MAPT P10636 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NR1H4 Q96RI1 1/20 0.39
LDLR P01130 1/20 0.37
PTPRC P08575 2/20 0.36
ESRRG P62508 2/20 0.36
KCNMA1 Q12791 2/20 0.35
CD274 Q9NZQ7 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
MDH1 P40925 1/20 0.35
MDH2 P40926 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9339491 0.92 HDAC1 (0.51) HDAC1F10PRSS1MAPTSMN1; SMN2
SCHEMBL9339500 0.85 ACHE (0.49) HDAC1F10PRSS1MAPTSMN1; SMN2
SCHEMBL9866208 0.83 BRD4 (0.44) HDAC1MAPTSMN1; SMN2NR1H4
SCHEMBL7307840 0.80 CA1 (0.46) PRSS1CD274
SCHEMBL9336123 0.78 ACHE (0.49) HDAC1F10PRSS1MAPTNR1H4
SCHEMBL9335835 0.78 BRD4 (0.45) HDAC1MAPTSMN1; SMN2NR1H4
SCHEMBL2659302 0.74 CD274 (0.56) HDAC1PRSS1MAPTSMN1; SMN2CD274
SCHEMBL7302006 0.74 SYK (0.46) PRSS1MAPTSMN1; SMN2
SCHEMBL9339289 0.73 MEN1 (0.43) HDAC1NR1H4
SCHEMBL8382918 0.73 ATM (0.48) HDAC1PRSS1MAPTNR1H4PTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5039805-A Novel benzoic and phenylacetic acid derivatives HOFFMANN-LA ROCHE INC. (US) 1991-08-13 US disclosed