SCHEMBL9866959

SCHEMBL9866959

COc1cc(NC(C)=O)c([N+](=O)[O-])cc1C(=O)NC1CCN(CC2CCCCC2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.56
MLNR O43193 1/20 0.52
ADRB2 P07550 1/20 0.52
CHRM1 P11229 1/20 0.52
DRD2 P14416 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
CHRM3 P20309 1/20 0.52
SLC6A2 P23975 1/20 0.52
HTR2A P28223 1/20 0.52
SLC6A4 P31645 1/20 0.52
HRH1 P35367 1/20 0.52
DRD3 P35462 1/20 0.52
OPRK1 P41145 1/20 0.52
HTR2B P41595 1/20 0.52
CHRNA4 P43681 1/20 0.52
HTR3A P46098 1/20 0.52
SLC6A3 Q01959 1/20 0.52
KCNH2 Q12809 1/20 0.52
HRH3 Q9Y5N1 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865507 0.89 DRD2 (0.67) DRD4MLNRADRB2CHRM1DRD2
SCHEMBL9868098 0.86 MLNR (0.65) MLNRADRB2CHRM1DRD2ADRA2B
SCHEMBL11549582 0.85 DRD4 (0.75) DRD4DRD2DRD3HTR4
Hydrochloric Acid SCHEMBL11548804 0.84 DRD4 (0.72) DRD4DRD2DRD3HTR4
Iodomethane SCHEMBL11548212 0.84 DRD4 (0.72) DRD4DRD2DRD3HTR4
SCHEMBL9867273 0.83 DRD4 (0.65) DRD4DRD2ADRA2BADRA2CSLC6A2
SCHEMBL9868673 0.83 DRD4 (0.51) DRD4DRD2ADRA2BADRA2CSLC6A2
SCHEMBL9867302 0.83 DRD4 (0.57) DRD4DRD2ADRA2BADRA2CSLC6A2
SCHEMBL9867056 0.83 DRD4 (0.55) DRD4DRD2ADRA2BADRA2CSLC6A2
SCHEMBL9867489 0.81 DRD4 (0.49) DRD4DRD2ADRA2BADRA2CSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5026858-A Used for treating nausea, vomating, gastrointestinal disorders and centarl nervous system WALTON S.A. (ES) 1991-06-25 US disclosed