SCHEMBL9867735

SCHEMBL9867735

CC(=O)c1c(O)ccc(C(C)(C)C)c1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.49
THRB P10828 1/20 0.48
GLRA3 O75311 1/20 0.47
GLRB P48167 1/20 0.47
CA2 P00918 1/20 0.45
ESRRA P11474 1/20 0.42
ALDH1A1 P00352 4/20 0.41
ALOX15 P16050 2/20 0.41
LMNA P02545 2/20 0.41
NR1I2 O75469 1/20 0.41
CYP2C9 P11712 1/20 0.41
MIF P14174 1/20 0.41
TYR P14679 1/20 0.41
HTT P42858 1/20 0.41
NFE2L2 Q16236 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CA9 Q16790 1/20 0.40
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
TDP1 Q9NUW8 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4122613 0.84 GLRA3 (0.62) GLRA3GLRBCA2ESRRAALDH1A1
SCHEMBL3630959 0.82 THRB (0.47) PRKCITHRBGLRA3GLRBCA2
SCHEMBL4122067 0.79 CA2 (0.55) GLRA3GLRBCA2ALDH1A1ALOX15
SCHEMBL1878648 0.78 THRB (0.61) PRKCITHRBCA2ALDH1A1HSD17B10
SCHEMBL6451162 0.75 THRB (0.70) PRKCITHRBCA2ALDH1A1ALOX15
SCHEMBL3185583 0.73 PRKCI (0.76) PRKCITHRBCA9GABRA1GABRB2
SCHEMBL3169896 0.73 CA2 (0.56) GLRA3GLRBCA2ALDH1A1ALOX15
SCHEMBL29488108 0.73 CA2 (0.56) GLRA3GLRBCA2ALDH1A1ALOX15
SCHEMBL9312650 0.72 THRB (0.54) PRKCITHRBALDH1A1ALOX15CYP2C9
SCHEMBL3280277 0.72 THRB (0.54) PRKCITHRBCA2ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006549-A Antiinflammatory agents MERCK & CO., INC. (US) 1991-04-09 US disclosed
EP-0399773-A1 Novel 7-aroyl-4-hydroxy-3-methyl benzolfurans as dual inhibitors of cyclooxygenase and 5-lipoxygenase MERCK & CO. INC. (US) 1990-11-28 EP disclosed
EP-0104018-A2 Benzopyran, benzothiapyran and quinoline compounds and pharmaceutical compositions containing them FISONS plc (GB) 1984-03-28 EP disclosed