SCHEMBL9869259

SCHEMBL9869259

COC(=O)c1cccnc1SCc1cccc(OC)c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.73
L3MBTL1 Q9Y468 1/20 0.73
KMT2A Q03164 4/20 0.54
MEN1 O00255 3/20 0.54
SMN1; SMN2 Q16637 5/20 0.52
MAPT P10636 3/20 0.52
HTT P42858 2/20 0.52
TDP1 Q9NUW8 2/20 0.52
ALDH1A1 P00352 4/20 0.52
CYP2C9 P11712 1/20 0.52
CYP1A2 P05177 1/20 0.51
HPGD P15428 3/20 0.51
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
POLB P06746 3/20 0.49
TP53 P04637 2/20 0.49
LMNA P02545 2/20 0.48
KDM4E B2RXH2 1/20 0.48
CDC7 O00311 1/20 0.47
DBF4 Q9UBU7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869842 0.89 KMT2A (0.68) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL8630241 0.85 L3MBTL1 (1.00) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL3421265 0.79 L3MBTL1 (0.79) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL4021262 0.77 KDR (0.64) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL4017666 0.75 L3MBTL1 (0.65) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL9661173 0.75 PKM (0.68) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL18795683 0.73 L3MBTL1 (0.64) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL13242893 0.73 L3MBTL1 (0.76) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL4018474 0.72 SMN1; SMN2 (0.65) PKML3MBTL1KMT2AMEN1SMN1; SMN2
SCHEMBL9661093 0.72 L3MBTL1 (0.71) PKML3MBTL1KMT2ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006532-A Enzyme inhibitor; antiinflammatory agents MERCK & CO. INC., INC. (US) 1991-04-09 US disclosed
US-4904672-A Derivatives of 3-hydroxyazabenzo[b]thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1990-02-27 US disclosed
US-4767766-A Derivatives of 3-hydroxyazabenzo(B)thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-08-30 US disclosed