SCHEMBL9869834

SCHEMBL9869834

Brc1ccc(-c2ccnc3nccn23)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.54
BACE1 P56817 2/20 0.46
EGLN2 Q96KS0 1/20 0.45
KDM4E B2RXH2 3/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
GAA P10253 3/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TP53 P04637 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ACVR1 Q04771 3/20 0.40
CHEK1 O14757 2/20 0.40
DYRK1A Q13627 2/20 0.40
MAP4K4 O95819 1/20 0.40
CSF1R P07333 1/20 0.40
PRKACA P17612 1/20 0.40
KDR P35968 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11009860 0.81 BACE1 (0.62) IDO1BACE1EGLN2NPC1RAB9A
SCHEMBL11010979 0.71 SMN1; SMN2 (0.58) BACE1EGLN2KDM4EGAAMAPT
SCHEMBL9869687 0.69 BACE1 (0.68) IDO1BACE1EGLN2KDM4EGAA
SCHEMBL9870329 0.67 TUBB4A (0.53) EGLN2KDM4EMAPTALDH1A1HPGD
SCHEMBL9870207 0.66 KDM4E (0.49) BACE1EGLN2KDM4EGAAMAPT
SCHEMBL25296092 0.64 BACE1 (0.70) BACE1KDM4ENPC1RAB9AGAA
SCHEMBL3036429 0.63 EGLN2 (0.49) BACE1EGLN2KDM4ERAB9AGAA
SCHEMBL6217374 0.63 EGLN2 (0.41) IDO1BACE1EGLN2ACVR1CHEK1
SCHEMBL2396066 0.63 EGLN2 (0.41) BACE1EGLN2RAB9AACVR1CHEK1
SCHEMBL7903223 0.63 EGLN2 (0.41) BACE1EGLN2ACVR1CHEK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5072042-A Skin disorders, anticarcinogenic-antitumor agent BASF AKTIENGESELLSCHAFT (DE) 1991-12-10 US claimed
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US disclosed