SCHEMBL9869687

SCHEMBL9869687

Clc1cccc(-c2ccnc3nccn23)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.68
EGLN2 Q96KS0 2/20 0.59
GAA P10253 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
IDO1 P14902 2/20 0.43
DYRK1A Q13627 2/20 0.42
DYRK1B Q9Y463 2/20 0.42
MAP4K4 O95819 2/20 0.42
KDR P35968 2/20 0.42
CHEK1 O14757 1/20 0.42
CSF1R P07333 1/20 0.42
PRKACA P17612 1/20 0.42
CDK8 P49336 1/20 0.42
MAP2K1 Q02750 1/20 0.42
ACVR1 Q04771 1/20 0.42
MAP4K2 Q12851 1/20 0.42
ROCK1 Q13464 1/20 0.42
AURKB Q96GD4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870207 0.77 KDM4E (0.49) BACE1EGLN2GAAKDM4EALDH1A1
SCHEMBL9869668 0.74 EGLN2 (1.00) BACE1EGLN2GAAKDM4EALDH1A1
SCHEMBL11010979 0.73 SMN1; SMN2 (0.58) BACE1EGLN2GAAKDM4EALDH1A1
SCHEMBL14920062 0.72 EGLN2 (0.68) BACE1EGLN2IDO1MAP2K1PIM1
SCHEMBL5462584 0.72 KDM4E (0.70) BACE1EGLN2GAAKDM4EALDH1A1
SCHEMBL11009860 0.72 BACE1 (0.62) BACE1EGLN2GAAALDH1A1SMN1; SMN2
SCHEMBL10474240 0.71 IKBKB (0.44) BACE1GAAKDM4EIDO1DYRK1A
Hydrochloric Acid SCHEMBL11014780 0.70 BACE1 (0.61) BACE1EGLN2GAAALDH1A1SMN1; SMN2
SCHEMBL9869834 0.69 IDO1 (0.54) BACE1EGLN2GAAKDM4EALDH1A1
SCHEMBL5408046 0.69 BACE1 (0.53) BACE1EGLN2KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US claimed
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US disclosed