SCHEMBL9870080

SCHEMBL9870080

CCNCC1CCN(c2c(F)cc3c(=O)c(C(=O)O)cn(-c4ccccc4)c3c2Cl)C1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
POLB P06746 1/20 0.51
CHRM2 P08172 1/20 0.51
CHRM1 P11229 1/20 0.51
OPRM1 P35372 1/20 0.51
OPRD1 P41143 1/20 0.51
TOP1 P11387 5/20 0.49
KDM4E B2RXH2 1/20 0.48
KCNH2 Q12809 1/20 0.47
TOP2A P11388 10/20 0.47
TOP2B Q02880 10/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10897095 0.93 KDM4E (0.55) ALDH1A1TOP1KDM4EKCNH2TOP2A
SCHEMBL11002445 0.91 TOP1 (0.44) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL10894425 0.87 TOP1 (0.51) ALDH1A1POLBTOP1KDM4EKCNH2
SCHEMBL10765111 0.86 ALDH1A1 (0.56) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL10530714 0.86 ALDH1A1 (0.70) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9869688 0.85 TOP1 (0.60) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL24334178 0.83 TOP1 (0.61) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL10893344 0.81 KCNH2 (0.62) ALDH1A1TOP1KDM4EKCNH2TOP2A
SCHEMBL10619519 0.81 KDM4E (0.53) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9869932 0.80 ALDH1A1 (0.62) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4981854-A BACTERICIDES, ANIMAL GROWTH REGUALTORS BAYER AKTIENGESELLSCHAFT (DE) 1991-01-01 US claimed
US-4980353-A BACTERICIDES, ANIMAL GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1990-12-25 US claimed
EP-0201829-A1 1-Aryl-4-quinolone-3-carboxylic acids BAYER AG (DE) 1986-11-20 EP claimed
US-4981854-A BACTERICIDES, ANIMAL GROWTH REGUALTORS BAYER AKTIENGESELLSCHAFT (DE) 1991-01-01 US disclosed
US-4980353-A BACTERICIDES, ANIMAL GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1990-12-25 US disclosed