SCHEMBL9870176

SCHEMBL9870176

CCN(CCC1CCCN1C)CC(=O)N1c2ccccc2C(=O)Nc2cccnc21

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 5/20 0.67
CHRM4 P08173 2/20 0.65
CHRM1 P11229 2/20 0.65
CHRM3 P20309 2/20 0.65
CYP1A2 P05177 1/20 0.65
CYP3A4 P08684 1/20 0.65
MAPK1 P28482 1/20 0.65
CHRM5 P08912 1/20 0.61
ALOX15 P16050 1/20 0.61
DRD1 P21728 1/20 0.61
DRD5 P21918 1/20 0.61
TMEM97 Q5BJF2 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871211 0.94 CHRM2 (0.59) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL8879790 0.90 CHRM2 (0.61) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL9870103 0.90 CHRM2 (0.54) CHRM2CHRM4CHRM1CHRM3CYP1A2
Hydrochloric Acid SCHEMBL9870848 0.90 CHRM2 (0.60) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL9871047 0.89 CHRM2 (0.58) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10459903 0.88 CHRM2 (0.62) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL8879186 0.87 CHRM2 (0.61) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10519813 0.85 CHRM2 (0.61) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10510299 0.84 CYP1A2 (0.85) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10515060 0.83 CHRM2 (0.71) CHRM2CHRM4CHRM1CHRM3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5002943-A Antispasmodic Agents, Bradycardia Treatment MIHM GERHARD (DE) 1991-03-26 US disclosed
EP-0346745-A1 Condensed diazepinones, processes for their preparation and pharmaceutical preparations containing them Dr. Karl Thomae GmbH (DE) 1989-12-20 EP disclosed
EP-0173462-B1 ELLIPTICINE DERIVATIVE AND PRODUCTION PROCESS THEREOF SUNTORY LIMITED (JP) 1989-10-25 EP disclosed