SCHEMBL9870468

SCHEMBL9870468

CC(C)(C)CC(=O)Oc1nn(Cc2cc3c(Cl)cccc3s2)c(=O)c2ncccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 8/20 0.50
SLC22A12 Q96S37 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33
KDM4E B2RXH2 2/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX12 P18054 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HTT P42858 2/20 0.33
MITF O75030 1/20 0.33
LMNA P02545 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870643 0.93 AKR1B1 (0.52) AKR1B1SLC22A12RXFP1KDM4EPDE4A
SCHEMBL9203840 0.82 AKR1B1 (0.56) AKR1B1KDM4EPDE4APDE4BPDE4C
SCHEMBL10431002 0.80 AKR1B1 (0.51) AKR1B1RXFP1KDM4EPDE4APDE4B
SCHEMBL9870061 0.78 AKR1B1 (0.77) AKR1B1
SCHEMBL9870702 0.75 AKR1B1 (0.54) AKR1B1
SCHEMBL9870079 0.75 AKR1B1 (0.36) AKR1B1RAB9ASMN1; SMN2
SCHEMBL9206507 0.74 AKR1B1 (0.77) AKR1B1
SCHEMBL9870810 0.74 AKR1B1 (0.67) AKR1B1
SCHEMBL10431004 0.74 AKR1B1 (0.57) AKR1B1KDM4EPDE4APDE4BPDE4C
SCHEMBL9870990 0.73 AKR1B1 (0.62) AKR1B1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4996204-A Antidiabetic agents PFIZER INC. (US) 1991-02-26 US disclosed