SCHEMBL9870683

SCHEMBL9870683

CCSc1ccc(N=C=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.42
TRPA1 O75762 1/20 0.40
SLC6A4 P31645 9/20 0.39
MAOA P21397 1/20 0.39
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 1/20 0.38
GSK3B P49841 1/20 0.36
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1899851 0.80 CYP3A4 (0.50) CYP3A4TSHRHSD17B10TRPA1GABRA1
SCHEMBL11646222 0.80 HSD17B10 (0.59) HSD17B10SLC6A4MAOAGABRA1GABRB2
SCHEMBL11531569 0.80 CYP3A4 (0.50) CYP3A4TSHRHSD17B10TRPA1GABRA1
Butane SCHEMBL16872374 0.78 CYP3A4 (0.62) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL2651634 0.78 GABRA1 (0.42) CYP3A4TSHRTRPA1SLC6A4MAOA
SCHEMBL546217 0.77 CYP3A4 (0.50) CYP3A4TSHRHSD17B10TRPA1SLC6A4
SCHEMBL11215338 0.77 CYP3A4 (0.43) CYP3A4TSHRHSD17B10TRPA1GABRA1
SCHEMBL739866 0.76 CYP3A4 (0.54) CYP3A4TSHRHSD17B10TRPA1GABRA1
SCHEMBL484003 0.76 CYP3A4 (0.54) CYP3A4TSHRHSD17B10TRPA1MAOA
SCHEMBL8870019 0.76 HSD17B10 (0.73) CYP3A4TSHRHSD17B10CYP1A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4996208-A Pesticidal thiazolopyrimidine derivatives BAYER AKTIENGESELLSCHAFT (DE) 1991-02-26 US disclosed
EP-0348746-A2 Thiazolopyrimidine derivatives, process for their preparation and their use as pest control agents BAYER AG (DE) 1990-01-03 EP disclosed
US-4174398-A Combating fungi with 1-alkyl-1-(1,3,4-thiadiazol-2-yl)-3-phenyl-ureas BAYER AKTIENGESELLSCHAFT (DE) 1979-11-13 US disclosed