SCHEMBL9870992

SCHEMBL9870992

O=C(Cl)c1ccc(OC(F)(F)C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
TRPV1 Q8NER1 6/20 0.38
EPHX2 P34913 3/20 0.38
TLR7 Q9NYK1 1/20 0.37
PPARA Q07869 2/20 0.37
FABP2 P12104 1/20 0.37
PPARG P37231 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
FAAH O00519 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9172265 0.87 ALDH1A1 (0.40) ALDH1A1TSHRHSD17B10NPC1RAB9A
SCHEMBL162647 0.84 EPHX2 (0.53) NPC1RAB9ATRPV1EPHX2TLR7
SCHEMBL1505766 0.83 ALDH1A1 (0.40) ALDH1A1TSHRHSD17B10NPC1RAB9A
SCHEMBL2715757 0.82 TSHR (0.59) ALDH1A1TSHRHSD17B10EPHX2FAAH
SCHEMBL9871408 0.82 ALDH1A1 (0.42) ALDH1A1TSHRHSD17B10NPC1RAB9A
SCHEMBL10910722 0.82 ALDH1A1 (0.47) ALDH1A1TSHRHSD17B10NPC1RAB9A
SCHEMBL2091503 0.81 MAPT (0.55) ALDH1A1TSHRHSD17B10RAB9AMAPT
SCHEMBL2091498 0.81 ALDH1A1 (0.41) ALDH1A1TSHRHSD17B10NPC1RAB9A
SCHEMBL9578494 0.79 HSD17B10 (0.48) ALDH1A1HSD17B10NPC1RAB9ATRPV1
SCHEMBL22815931 0.79 AURKA (0.54) NPC1RAB9ATRPV1EPHX2TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047584-A Process for the preparation of pentahaloethoxy benzoyl halide compounds OCCIDENTAL CHEMICAL CORP. (US) 1991-09-10 US disclosed
EP-0002906-B1 NOVEL PERIMIDINES, THEIR PREPARATION, FORMULATIONS AND USE AS IMMUNOSUPPRESSIVES ELI LILLY AND COMPANY (US) 1982-04-14 EP disclosed
US-4294964-A IMMUNOSUPRESSIVE AGENTS ELI LILLY AND COMPANY (US) 1981-10-13 US disclosed
US-4224326-A 2-ARYL-1H-PERIMIDINES ELI LILLY AND COMPANY (US) 1980-09-23 US disclosed
EP-0002906-A2 Novel perimidines, their preparation, formulations and use as immunosuppressives ELI LILLY AND COMPANY (US) 1979-07-11 EP disclosed
US-3960945-A 4-[-(Alkoxy or polyhaloalkoxy)-benzamido]cyclohexanones STERLING DRUG INC. (US) 1976-06-01 US disclosed