SCHEMBL9871014

SCHEMBL9871014

Cc1nccc(-c2ccccc2)c1C=CC(O)CC(=O)CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.38
HMGCR P04035 3/20 0.36
MMP12 P39900 1/20 0.35
CTSA P10619 2/20 0.35
CASP1 P29466 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
GPR119 Q8TDV5 1/20 0.33
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
ESR1 P03372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871007 1.00 TACR1 (0.38) TACR1HMGCRMMP12CTSACASP1
SCHEMBL9871610 0.88 ALDH1A1 (0.39) MEN1ALDH1A1KMT2AGPR119HPGD
SCHEMBL9871601 0.88 ALDH1A1 (0.39) MEN1ALDH1A1KMT2AGPR119HPGD
SCHEMBL10466197 0.83 HMGCR (0.46) HMGCRESR1
SCHEMBL9870912 0.83 HMGCR (0.46) HMGCRESR1
SCHEMBL10466201 0.83 HMGCR (0.46) HMGCRESR1
SCHEMBL9871615 0.81 HMGCR (0.35) TACR1HMGCRKMT2AGPR119NPC1
SCHEMBL8953313 0.79 HMGCR (0.49) HMGCR
SCHEMBL8953297 0.79 HMGCR (0.49) HMGCR
SCHEMBL9870230 0.77 HMGCR (0.43) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
EP-0306929-A2 6-[[(Substituted)pyridin-3-YL]alkyl]-and alkenyl]-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1989-03-15 EP disclosed