SCHEMBL9871601

SCHEMBL9871601

CCOC(=O)CC(=O)CC(O)/C=C/c1c(-c2ccccc2)ccnc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 4/20 0.39
HPGD P15428 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
NCOA1 Q15788 2/20 0.39
NCOA3 Q9Y6Q9 2/20 0.39
GPR119 Q8TDV5 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
PTPN1 P18031 1/20 0.37
HTT P42858 2/20 0.37
HSD17B10 Q99714 2/20 0.37
GRM4 Q14833 1/20 0.36
SQOR Q9Y6N5 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871610 1.00 ALDH1A1 (0.39) ALDH1A1KDM4EHPGDSMN1; SMN2MEN1
SCHEMBL9871014 0.88 TACR1 (0.38) ALDH1A1HPGDMEN1KMT2AGPR119
SCHEMBL9871007 0.88 TACR1 (0.38) ALDH1A1HPGDMEN1KMT2AGPR119
SCHEMBL9870230 0.85 HMGCR (0.43) PTPN1
SCHEMBL9871615 0.79 HMGCR (0.35) HPGDKMT2AGPR119
SCHEMBL10466201 0.77 HMGCR (0.46) ADORA3CYP2C9
SCHEMBL9870912 0.77 HMGCR (0.46) ADORA3CYP2C9
SCHEMBL10466197 0.77 HMGCR (0.46) ADORA3CYP2C9
SCHEMBL9420583 0.70 CNR2 (0.41) ALDH1A1LMNACYP1A2
SCHEMBL9420580 0.70 CNR2 (0.41) ALDH1A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed