SCHEMBL9871200

SCHEMBL9871200

Cc1nccc(-c2ccccc2)c1C=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.42
ERN1 O75460 2/20 0.40
PSMB5 P28074 1/20 0.39
GRM4 Q14833 1/20 0.39
HTT P42858 1/20 0.39
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
DAPK3 O43293 1/20 0.39
JAK2 O60674 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
PAK4 O96013 1/20 0.39
CSF1R P07333 1/20 0.39
RET P07949 1/20 0.39
IGF1R P08069 1/20 0.39
FGFR1 P11362 1/20 0.39
PRKACA P17612 1/20 0.39
FLT1 P17948 1/20 0.39
LTK P29376 1/20 0.39
GRK5 P34947 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871401 0.86 MEN1 (0.44) CHEK1GRM4IKBKBCHUKDAPK3
SCHEMBL9871387 0.86 MEN1 (0.44) CHEK1GRM4IKBKBCHUKDAPK3
SCHEMBL8846070 0.81 CHEK1 (0.42) CHEK1PSMB5GRM4IKBKBCHUK
SCHEMBL28198595 0.81 LRRK2 (0.39) CHEK1ERN1IKBKBCHUKDAPK3
SCHEMBL8550487 0.81 MEN1 (0.39) CHEK1IKBKBCHUKDAPK3JAK2
SCHEMBL25120727 0.81 RPS6KA3 (0.39) CHEK1IKBKBCHUKDAPK3JAK2
SCHEMBL30319423 0.81 RPS6KA3 (0.39) CHEK1IKBKBCHUKDAPK3JAK2
SCHEMBL22476115 0.80 MTOR (0.48) MAP4K4PRKACACDK9CLK4CYP17A1
SCHEMBL9871811 0.80 HCAR2 (0.43) CHEK1CDK8TACR1MEN1RAB9A
SCHEMBL9871808 0.80 HCAR2 (0.43) CHEK1CDK8TACR1MEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
EP-0306929-A2 6-[[(Substituted)pyridin-3-YL]alkyl]-and alkenyl]-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1989-03-15 EP disclosed