SCHEMBL9871401

SCHEMBL9871401

Cc1nccc(-c2ccccc2)c1C=CC=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
NPC1 O15118 2/20 0.44
POLB P06746 1/20 0.44
ALDH1A1 P00352 2/20 0.42
TRPA1 O75762 1/20 0.42
LMNA P02545 1/20 0.42
ALOX5 P09917 1/20 0.42
MAPK1 P28482 1/20 0.42
CHEK1 O14757 1/20 0.41
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
GRM4 Q14833 1/20 0.37
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
DAPK3 O43293 1/20 0.37
JAK2 O60674 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37
PAK4 O96013 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871387 1.00 MEN1 (0.44) MEN1KMT2ANPC1POLBALDH1A1
SCHEMBL9871200 0.86 CHEK1 (0.42) MEN1KMT2AALDH1A1LMNACHEK1
SCHEMBL9871811 0.80 HCAR2 (0.43) MEN1KMT2ANPC1POLBALDH1A1
SCHEMBL9871808 0.80 HCAR2 (0.43) MEN1KMT2ANPC1POLBALDH1A1
SCHEMBL8846070 0.79 CHEK1 (0.42) MEN1KMT2ANPC1ALDH1A1CHEK1
SCHEMBL9870737 0.78 CHEK1 (0.40) MEN1KMT2ANPC1ALDH1A1CHEK1
SCHEMBL9870731 0.78 CHEK1 (0.40) MEN1KMT2ANPC1ALDH1A1CHEK1
SCHEMBL18433892 0.76 CYP17A1 (0.43) MEN1KMT2AALDH1A1LMNACHEK1
SCHEMBL9871017 0.75 KMT2A (0.43) MEN1KMT2AALDH1A1ALOX5CDK8
SCHEMBL9871013 0.75 KMT2A (0.43) MEN1KMT2AALDH1A1ALOX5CDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed