SCHEMBL9871808

SCHEMBL9871808

Cc1nccc(-c2ccccc2)c1/C=C/C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.43
HDAC3 O15379 1/20 0.43
TNKS O95271 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
TACR1 P25103 2/20 0.42
ALDH1A1 P00352 5/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
HPGD P15428 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871811 1.00 HCAR2 (0.43) HCAR2HDAC3TNKSHDAC4HDAC1
SCHEMBL9871013 0.85 KMT2A (0.43) HDAC3HDAC1HDAC8TACR1ALDH1A1
SCHEMBL9871017 0.85 KMT2A (0.43) HDAC3HDAC1HDAC8TACR1ALDH1A1
SCHEMBL9871401 0.80 MEN1 (0.44) TACR1ALDH1A1GAASMN1; SMN2POLB
SCHEMBL9871387 0.80 MEN1 (0.44) TACR1ALDH1A1GAASMN1; SMN2POLB
SCHEMBL9871200 0.80 CHEK1 (0.42) TACR1ALDH1A1MEN1KMT2AMKNK1
SCHEMBL9870737 0.79 CHEK1 (0.40) TACR1ALDH1A1SMN1; SMN2L3MBTL1MEN1
SCHEMBL9870731 0.79 CHEK1 (0.40) TACR1ALDH1A1SMN1; SMN2L3MBTL1MEN1
SCHEMBL9871009 0.78 AKR1C3 (0.46) TACR1RXRARXRBNR4A2MKNK1
SCHEMBL9871020 0.78 AKR1C3 (0.46) TACR1RXRARXRBNR4A2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
EP-0306929-A2 6-[[(Substituted)pyridin-3-YL]alkyl]-and alkenyl]-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1989-03-15 EP disclosed